GSK1016790A is supplied by Merck (Sigma-Aldrich). It is utilized:

to stimulate transient receptor potential vanilloid 4 (TRPV4)-mediated currents in Xenopus laevis oocytes

to stimulate cells in Ca2+ level measurement in human retinal capillary endothelial cells (HRCECs)

to study the role of TRPV4 channels in brain injury after intracerebral hemorrhage (ICH)

to trigger the opening of TRPV4 channels in bovine nucleus pulposus cells or Hanks Balanced Salt Solution

PRODUCT SPECIFICATIONS:

Name: GSK1016790A

Brand: Merck (Sigma-Aldrich)

Pack size: 5MG

Catalog number: P0122-5MG

PRODUCT FEATURES:

Synonym: (N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide, GSK101

CAS Number: 942206-85-1

Empirical Formula: C28H32Cl2N4O6S2

Molecular Weight: 655.61